Table 3:
Aminosalicylates, Doses, and Intestinal Activity
Medication
Dosage
Colon Activity
Small-bowel activity
Distal
Proximal
Sulfasalazine
2-8 g/d
++
+++
-
Olsalazine
1-3 g/d
++
+++
-
Balsalzide
6.75-12 g/d
+++
+++
-
Pentasa ® (melsalamine)
2-4 g/d
++
++
++
Asacol ® (mesalamine)
2.4-4.8 g/d
++
+++
+
Rowasa enemas ®
(mesalamine)
4 g/d
+++
-
-
Canasa suppositories™
(mesalamine)
2-4 g/d
+
-
-
  
Copyright 2002 The Cleveland Clinic Foundation

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