Table 3:
Aminosalicylates, Doses, and Intestinal Activity
Medication
Dosage
Colon Activity
Small-bowel activity
Distal
Proximal
Sulfasalazine
2-8 g/d
++
+++
-
Olsalazine
1-3 g/d
++
+++
-
Balsalzide
6.75-12 g/d
+++
+++
-
Pentasa
®
(melsalamine)
2-4 g/d
++
++
++
Asacol
®
(mesalamine)
2.4-4.8 g/d
++
+++
+
Rowasa enemas
®
(mesalamine)
4 g/d
+++
-
-
Canasa suppositories
(mesalamine)
2-4 g/d
+
-
-
Copyright 2002 The Cleveland Clinic Foundation
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